Clipos™ A939572 Encapsulated Liposomes


Catalog:CDEPG-27

Unit Size:2 mL, 10 mL

INQUIRY Datasheet

Specifications
Description PEGylated liposomes containing SCD1 inhibitor A939572. A939572 is a potent stearoyl-CoA desaturase 1 (SCD1) inhibitor with reported IC50s of <4 nM and 37 nM for mouse and human SCD1, respectively. A939572 is insoluble in aqueous media. This product is a pre-formulated liposomal version of A939572 which is supplied ready to use in vitro or in vivo. The liposomes are PEGylated for optimal in vivo performance. For preclinical research use only.
Lipid composition PEGylated Liposomes
Liposome Size 70-120 nm
Lipid Molar Concentration 60 mM
Encapsulated Drug A939572
Drug concentration 500 mcg/mL
Inside Buffer 292 mM sucrose, 0.5% DPBS (1X)
Outside Buffer 292 mM sucrose, 0.5% DPBS (1X)
Storage 2 °C to 8 °C (do not freeze), protect from light
Shelf-life At least 1 month
CAS No. 1032229-33-6
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