Clipos™ Belinostat (PXD101) Encapsulated Liposomes


Catalog:CDEPG-33

Unit Size:2 mL, 10 mL

INQUIRY Datasheet

Specifications
Description PEGylated liposomes containing HDAC inhibitor Belinostat (PXD101, NSC726630, PX-105684). Belinostat is a histone deacetylase inhibitor (HDACi) with reported IC50 of 27 nM (cell-free assay) and has been reported to induce autophagy and possess activity in cisplatin-resistant tumors. The liposomes are PEGylated for optimal in vivo performance. For preclinical research use only.
Lipid composition PEGylated Liposomes
Liposome Size 70-120 nm
Lipid Molar Concentration 60 mM
Encapsulated Drug Belinostat (PXD101, NSC726630, PX-105684)
Drug concentration 3.1 mg/mL
Inside Buffer 292 mM sucrose, 0.5% DPBS (1X)
Outside Buffer 292 mM sucrose, 0.5% DPBS (1X)
Storage 2 °C to 8 °C (do not freeze)
Shelf-life 1 month
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