Clipos™ Mirdametinib (PD0325901) Encapsulated Liposomes


Catalog:CDEPG-32

Unit Size:1mL, 2.5 mL, 5mL, 10 mL

INQUIRY Datasheet

Specifications
Description PEGylated liposomes containing MEK inhibitor Mirdametinib (PD0325901). Mirdametinib (PD0325901) is a selective and non ATP-competitive MEK inhibitor with an IC50 of 0.33 nM (cell-free assays). The liposomes are PEGylated for optimal in vivo performance. For preclinical research use only.
Lipid composition PEGylated Liposomes
Liposome Size 70-120 nm
Lipid Molar Concentration 60 mM
Encapsulated Drug Mirdametinib PD0325901
Drug concentration 10.0 mg/mL (± ~5%)
Inside Buffer 292 mM sucrose, 0.5% DPBS (1X)
Outside Buffer 292 mM sucrose, 0.5% DPBS (1X)
Storage 2 °C to 8 °C (do not freeze)
Shelf-life 3 months
CAS No. 391210-10-9
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